Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ UCN-01
A cell-permeable Staurosporine derived anticancer agent that reversibly and ATP-competitively inhibits several protein kinases.
MilliporeSigma™ Calbiochem™ GGTI-286
A potent, cell-permeable, and selective inhibitor of GGTase I.
MilliporeSigma™ Calbiochem™ PP1 Analog III, 3-MB-PP1
PP1 Analog III, 3-MB-PP1 primarily used in Inhibition.
MilliporeSigma™ Calbiochem™ IKK Inhibitor III, BMS-345541
IKK Inhibitor III, BMS-345541, CAS 445430-58-0, is a cell-permeable, potent, selective, and allosteric site-binding inhibitor of IKK-2 (IC50 = ≈300 nM).
MilliporeSigma™ Calbiochem™ Caspase-9 Inhibitor III
The Caspase-9 Inhibitor III, also referenced under CAS 403848-57-7, controls the biological activity of Caspase-9. This small molecule/inhibitor is primarily used for Cancer applications.
MilliporeSigma™ Calbiochem™ Gö 6983
A potent, cell-permeable, reversible, and ATP-competitive inhibitor of protein kinase C (PKC) that inhibits several PKC isozymes.
MilliporeSigma™ Calbiochem™ Batimastat
Batimastat primarily used in Inhibition.
MilliporeSigma™ Calbiochem™ Interleukin-1 Receptor-Associated-Kinase-1/4 Inhibitor
The Interleukin-1 Receptor-Associated-Kinase-1/4 Inhibitor controls the activity of Interleukin-1 Receptor-Associated-Kinase-1/4. Primarily used for Phosphorylation & Dephosphorylation apps.
MilliporeSigma™ Calbiochem™ Protease Inhibitor Cocktail Set II
The Protease Inhibitor Cocktail Set II controls the activity of Protease. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ InSolution™ PERK Inhibitor I, GSK2606414
A cell-permeable pyrrolopyrimidinamine compound that acts as a highly potent inhibitor against EIF2AK3/PERK-catalyzed EIF2α Ser51 phosphorylation in kinase assays (IC50 = 0
MilliporeSigma™ Calbiochem™ Hh Signaling Antagonist X, Itraconazole
The Hh Signaling Antagonist X, Itraconazole, also referenced under CAS 84625-61-6, controls the biological activity of Hh pathway. This small molecule/inhibitor is primarily used for Cell Signaling applications.
MilliporeSigma™ Calbiochem™ Benztropine
An antagonist of muscarinic M1 and M3 receptors that induces robust differentiation of oligodendrocytes precursor cell differentiation (EC50 = 500nM) and promotes myelination.
MilliporeSigma™ Calbiochem™ Pepstatin A, Penetratin
A Pepstatin A that is ≈75% less potent against Cathespins D/E than PepA in cell-free assays.
MilliporeSigma™ Calbiochem™ HBDDE
A cell-permeable protein kinase C (PKC) inhibitor that selectively inhibits PKCα and PKCγ over PKCδ, βI, and βII isozymes in in vitro assays.
MilliporeSigma™ Calbiochem™ Proteasome Inhibitor Set II
The Proteasome Inhibitor Set II controls the biological activity of Proteasome. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.